Evidence-based peptide information for research and educational purposes only.
GH Secretagogues
Protocol not independently verified GH Axis Repair
Educational reference only. Read the full disclaimer. The protocols below are not automatically an FDA-approved or clinically verified regimen unless explicitly marked as label-verified or human-trial protocol above.

Overview

Route(s): Subcutaneous

Typical vial sizes: 1 mg

Dosing window: Post-Workout

Receptor / target: IGF-1

Properties: Not stated

Pre-mixed: No

Protocol examples

Standard Protocol

TimeframeDoseNotes
Week 133mcg daily1x/day, 7 days per week. Dose immediately post-workout (within 30 mins) with carbs and protein.
Week 250mcg daily1x/day, 7 days per week. Avoid taking at bedtime or while fasted.
Weeks 3-475mcg daily1x/day, 7 days per week. Ensure adequate calories/protein are consumed.
Weeks 5-8100mcg daily1x/day, 7 days per week. Maximum recommended dosage phase.

Protocol example from the source dataset; verify against the evidence status and listed sources.

Alternative: Bilateral IM

TimeframeDoseNotes
Weeks 1-850mcg split (25mcg per side)Administered intramuscularly into the trained muscle group (e.g., left and right bicep) immediately post-workout.

Alternative example from the source dataset; not an approved-label regimen unless marked above.

Protocol logic check

Protocol context: GH-axis protocols are not 'more is better.' The logic is pulse quality, recovery time, IGF-1/glucose monitoring, and avoiding receptor desensitization, edema, appetite spikes, numbness, or blood-pressure strain. Entry context: target (IGF-1); route Subcutaneous; timing Post-Workout. Unapproved or source-dataset dosing tables are hypotheses, not recommendations.

Independent evidence

Independent safety notes: No approved-label regimen was identified for this entry. Dosing examples should be treated as unverified protocol examples.

Regulatory status: no approved label identified

Storage

No approved-label storage guidance was identified for this entry. Use conservative sterile handling and see the general storage guidance in the FAQ.

Contraindications & cautions

Evidence varies by item. Some points come from labels, published literature, or regulatory context; others are mechanism-based cautions from the source dataset. Use the sources below to verify details.

  • Active cancer: IGF-1 is a potent mitogen; direct IGF-1 receptor activation accelerates proliferation of malignant cells.
  • History of malignancy: especially hormone-sensitive cancers; IGF-1 receptor signaling drives tumor growth in breast, prostate, and colorectal cancers.
  • Hypoglycemia or hypoglycemia unawareness: acute hypoglycemia is the primary risk; IGF-1 receptor activity mimics insulin; never administer fasted.
  • Diabetic ketoacidosis.
  • Type 1 or insulin-dependent diabetes: IGF-1's insulin-like activity requires careful glycemic management.
  • Concurrent use with insulin: severe additive hypoglycemia risk; extreme caution required.
  • Concurrent administration without food: administration without concurrent carbohydrates and protein is contraindicated; hypoglycemia risk is immediate.
  • Pre-existing visceral organ enlargement: IGF-1 at high doses drives growth in all IGF-1 receptor-expressing tissues, including intestinal epithelium and visceral organs.
  • Active acromegaly: additive IGF-1 receptor stimulation in a state of existing IGF-1 excess.
  • Pregnancy: IGF-1 analog activity not established in pregnancy; potential fetal risk.
  • Breastfeeding: safety not established.
  • Known hypersensitivity to IGF-1 LR3 or excipients.
  • Pediatric use: safety and efficacy not established; open growth plates in children risk inappropriate and disproportionate skeletal growth.

Possible side effects

Evidence varies by item. Some points come from labels, published literature, or regulatory context; others are mechanism-based cautions from the source dataset. Use the sources below to verify details.

  • Severe hypoglycemia: the most critical adverse effect; direct insulin-like glucose uptake via IGF-1 receptor activation; onset typically 30-60 minutes post-injection; more pronounced with fasted administration; always administer with carbohydrates present.
  • Intestinal growth and gut hypertrophy: with abused long-term or excessive dosing, IGF-1 receptor stimulation in gastrointestinal epithelium can cause measurable organ enlargement; this is the primary long-term misuse risk.
  • Visceral organ growth: liver, spleen, kidneys; IGF-1 receptor is expressed in all visceral organs; supraphysiologic IGF-1 exposure over extended periods may drive size increases.
  • Localized swelling at injection site: tissue response to subcutaneous or intramuscular injection.
  • Edema: IGF-1-mediated sodium and fluid retention.
  • Jaw tightening or facial growth (at high doses/extended abuse): IGF-1 receptors in craniofacial tissues; acromegalic-type effects at very high doses.
  • Joint pain: GH/IGF-1 axis-mediated periarticular fluid.
  • Headache.
  • Fatigue: transient post-injection.
  • Nausea: dose-dependent.
  • Increased appetite: orexigenic effect of IGF-1 receptor activity.
  • Tingling or numbness in extremities: insulin-like effects and fluid shifts.
  • Carpal tunnel syndrome risk: with extended high-dose use.
  • Downregulation of endogenous GH production: negative feedback from elevated IGF-1 on hypothalamic-pituitary axis; natural GH production suppressed during and after long cycles.

Compatibility

The relationships below come from the source site's internal engine and were not verified independently. Treat them as a starting point for a conversation with a clinician. They carry no safety guarantee.

Reported synergistic:

Reported contraindicated combinations:

None listed.

Sources